Mocetinostat
Information
- Drug Name
- Mocetinostat
- Description
- Entry(CIViC)
- 1
CIViC
Disease | Mutation | EL | ET | ED | CS | VO | TR | Pubmed | Links |
---|---|---|---|---|---|---|---|---|---|
malignant mesothelioma | BAP1 MUTATION BAP1 MUTATION | E |
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Sensitivity/Response | Somatic | 2 | 25970771 | Detail |
Annotation
Description | Associated Genes | Associated Variants | Sensitivity | Supported | Source | Links |
---|---|---|---|---|---|---|
A siRNA screen identified BAP1 associated with HDA... | BAP1 | BAP1 MUTATION BAP1 MUTATION | Sensitivity | true | CIViC Evidence | detail |
NCT ID | Status | Phase | Summary | Start date | Completion date |
---|---|---|---|---|---|
NCT03220477 | Active, not recruiting | Phase 1 | Pembrolizumab (Immunotherapy Drug) in Combination With Guadecitabine and Mocetinostat (Epigenetic Drugs) for Patients With Advanced Lung Cancer. | August 4, 2017 | July 2024 |
NCT02236195 | Completed | Phase 2 | Study of Mocetinostat in Patients With Urothelial Carcinoma Having Inactivating Alterations of Specific Genes | October 2014 | July 2016 |
NCT02018926 | Completed | Phase 1/Phase 2 | Safety Study of Mocetinostat in Combination With Azacitidine in Subjects With MDS | December 2013 | September 2015 |
NCT02303262 | Completed | Phase 2 | SARC018: A Study of Mocetinostat and Gemcitabine in Patients With Metastatic Leiomyosarcoma | November 12, 2015 | December 2016 |
NCT04299113 | Recruiting | Phase 1 | Mocetinostat With Vinorelbine in Children, Adolescents & Young Adults With Refractory and/or Recurrent Rhabdomyosarcoma | May 14, 2020 | May 22, 2026 |
NCT02954991 | Terminated | Phase 2 | Phase 2 Study of Glesatinib, Sitravatinib or Mocetinostat in Combination With Nivolumab in Non-Small Cell Lung Cancer | November 7, 2016 | November 4, 2021 |
NCT02282358 | Terminated | Phase 1/Phase 2 | Study of Mocetinostat in Selected Patients With Mutations of Acetyltransferase Genes in Relapsed and Refractory Diffuse Large B-Cell Lymphoma and Follicular Lymphoma | October 2014 | May 26, 2023 |
NCT02993991 | Withdrawn | Phase 1 | Pre-operative Mocetinostat (MGCD0103) and Durvalumab (MEDI4736) (PRIMED) for Squamous Cell Carcinoma of the Oral Cavity | October 10, 2017 | December 21, 2017 |
- Target (Drug list of Screening Committee of Anticancer Drugs)
- Histone deacetylases (HDAC)
- Synonym (Drug list of Screening Committee of Anticancer Drugs)
- MGCD0103