Annotation Detail

Information
Associated Genes
MAP2K1
Associated Variants
MAP2K1 UNKNOWN
Source Database
MMMP
Description
CI-1040 is a MEK inhibitor
MMMP State
mut V211D
MMMP Molecule
MEK1
MMMP Relationship
resistance to
MMMP Drug
CI-1040
MMMP Drug Alias
PD184352
MMMP Model
3
MMMP Reference
Emery CM, Proc Natl Acad Sci USA 2009, 106:20411-6
MMMP DNA/mRNA/Protein
DNA
Drugs
Drug NameSensitivitySupported
CI-1040Resitance or Non-Reponsetrue