Annotation Detail
Information
- Associated Genes
- RAF1
- Associated Variants
- RAF1 EXPRESSION
- Source Database
- MMMP
- Description
- Melanoma cells expressing no ectopic C-Raf were more resistant to Sorafenib. Both oncogenic Ras and Sorafenib stabilize B-Raf(V600E)-C-Raf complexes, thereby impairing MAPK activation. This inhibitory function of C-Raf on B-Raf(V600E)-mediated MAPK activation may explain the lack of co-occurrence of B-Raf(V600E) and oncogenic Ras mutations
- MMMP State
- expressed
- MMMP Molecule
- CRAF
- MMMP Molecule Alias
- C-Raf
- MMMP Relationship
- sensitivity to
- MMMP Drug
- Sorafenib
- MMMP Drug Alias
- Nexavar (R)
- MMMP Model
- 3
- MMMP Reference
- Karreth FA, Mol Cell 2009, 36:477-86
- MMMP DNA/mRNA/Protein
- protein
Drugs
Drug Name | Sensitivity | Supported |
---|---|---|
Sorafenib | Sensitivity | true |