Annotation Detail

Information
Associated Genes
ABL1
Associated Variants
ABL1 BCR-ABL
Associated Disease
chronic myeloid leukemia
Source Database
CIViC Evidence
Description
The use of nilotinib and dasatinib, second-generation BCR-ABL targeted therapies, has been effective in patients resistant to imatinib, leading to their FDA-approval.
Variant Origin
somatic
Variant Origin
Somatic
Evidence URL
https://civic.genome.wustl.edu/links/evidence_items/261
Gene URL
https://civic.genome.wustl.edu/links/genes/4
Variant URL
https://civic.genome.wustl.edu/links/variants/1
Rating
4
Evidence Type
Predictive
Disease
Chronic Myeloid Leukemia
Evidence Direction
Supports
Drug
Dasatinib,Nilotinib
Evidence Level
A
Clinical Significance
Sensitivity/Response
Pubmed
20537386
Drugs
Drug NameSensitivitySupported
DasatinibSensitivitytrue
NilotinibSensitivitytrue