Annotation Detail
Information
- Associated Genes
- CDKN2A
- Associated Variants
-
CDKN2A LOSS
(
ENST00000579755.2 )
CDKN2A LOSS ( ENST00000579755.2 ) - Associated Disease
- dermatofibrosarcoma protuberans
- Source Database
- CIViC Evidence
- Description
- An imatinib-resistant cell line, DFSP105, was established from a dermatofibrosarcoma protuberans which had progressed to a high-grade fibrosarcomatous DFSP. The disease-associated PDGFB-COL1A1 fusion was consistent with the most common form, a supernumerary ring chromosome. Genetic characterization of the cell line with a SNP array identified a homozygous CDKN2A/B deletion. Treatment of this cell line with CDK4/6 inhibitor palbociclib led to growth inhibition and reduced RB1 phosphorylation in vitro and in-vivo.
- Variant Origin
- Unknown
- Variant Origin
- Unknown
- Evidence URL
- https://civic.genome.wustl.edu/links/evidence_items/1881
- Gene URL
- https://civic.genome.wustl.edu/links/genes/14
- Variant URL
- https://civic.genome.wustl.edu/links/variants/554
- Rating
- 2
- Evidence Type
- Predictive
- Disease
- Dermatofibrosarcoma Protuberans
- Evidence Direction
- Supports
- Drug
- Palbociclib
- Evidence Level
- D
- Clinical Significance
- Sensitivity/Response
- Pubmed
- 25852058
Drugs
Drug Name | Sensitivity | Supported |
---|---|---|
Palbociclib | Sensitivity | true |